tbResList Print — Vem verapamil

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Product

Vem verapamil
Description: <b>Verapamil</b> belongs to the phenylalkylamine class of compounds and is a fully synthetic molecule originally developed for its potent calcium channel–blocking properties.<br>
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Pathways:<br>
-P-glycoprotein Inhibition (MDR1). -P-gp is overexpressed in many cancer cells<br>
-Inhibition of P-gp by verapamil can enhance the intracellular concentration of chemotherapeutic agents, potentially restoring drug sensitivity.<br>
-As a calcium channel blocker, verapamil inhibits L-type calcium channels.<br>

Pathway results for Effect on Cancer / Diseased Cells

Redox & Oxidative Stress

ROS↑, 1,  

Cell Death

Casp↑, 1,   Proteasome↓, 1,  

Protein Folding & ER Stress

ER Stress↑, 1,  

Drug Metabolism & Resistance

eff↑, 2,  
Total Targets: 5

Pathway results for Effect on Normal Cells

Total Targets: 0

Research papers

Year Title Authors PMID Link Flag
2014Calcium channel blocker verapamil accelerates gambogic acid-induced cytotoxicity via enhancing proteasome inhibition and ROS generationNingning Liu24373880https://pubmed.ncbi.nlm.nih.gov/24373880/0